Stereoselective Synthesis, Crystal Structure and Fungicidal Activity oftrans-2,3,6(8)-Trisubstituted-1,3-benzoxazines
نویسندگان
چکیده
منابع مشابه
Synthesis and fungicidal activity of novel 2,3-disubstituted-1,3-benzoxazines.
A series of new 2,3-disubstituted-3,4-dihydro-2H-1,3-benzoxazines were prepared in moderate to excellent yields by aza-acetalizations of aromatic aldehydes with 2-(N-substituted aminomethyl)phenols in the presence of TMSCl. Their structures were confirmed by IR, ¹H-NMR, ¹³C-NMR, MS and elemental analysis. The fungicidal activities of the target compounds were preliminarily evaluated, and some c...
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ژورنال
عنوان ژورنال: Chinese Journal of Organic Chemistry
سال: 2016
ISSN: 0253-2786
DOI: 10.6023/cjoc201508019